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GW 4064

¥0
货号
2473
CAS 号
[278779-30-9]
分子式
C 28 H 22 Cl 3 NO 4
分子量
542.84
规格
10mg; 50mg
规格(数值)
10 mg
别名
3-[2-[2-Chloro-4-[[3-(2,6-dichlorop henyl)-5-(1-methylethyl)-4-isoxazolyl]methoxy]phen yl]ethenyl]benzoic acid
溶解性
Soluble to 100 mM in DMSO and to 10 mM in ethanol
储存条件
+4°C
销量
0

产品描述

Selective, non-steroidal farnesoid X receptor (FXR) agonist (EC 50 = 15 nM). Displays no activity at other nuclear receptors at concentrations up to 1 μM. Improves hyperglycaemia and hyperlipidemia in diabetic db/db mice. Purity: >97 %

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