XCT 790
¥0
- 货号
- XCT 790
- CAS 号
- [725247-18-7]
- 分子式
- C 23 H 13 F 9 N 4 O 3 S
- 分子量
- 596.42
- 规格
- 10mg; 50mg
- 规格(数值)
- 10 mg
- 别名
- 3-[4-(2,4-Bis-trifluoromethylbenzyl oxy)-3-methoxyphenyl]-2-cyano-N-(5-trifluoromethyl -1,3,4-thiadiazol-2-yl)acrylamide
- 溶解性
- Soluble to 25 mM in DMSO
- 储存条件
- Store at +4°C
- 销量
- 0
产品描述
Selective ERRα antagonist/inverse agonist (IC 50 = ~400 nM). Displays no antagonist activity at ERRγ or ERα at concentrations below 10 μM. Interferes with PPARγ coactivator-1α (PGC-1α)/ERRα-dependent signaling: inhibits PGC-1α induction of ERRα and MAO-B gene expression and downregulates the constitutive transcriptional activity of ERRα in numerous cell lines. Purity: >99 %