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Xanomeline oxalate

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货号
Xanomeline oxalate
CAS 号
[141064-23-5]
分子式
C 14 H 23 N 3 OS.C 2 H 2 O 4
分子量
371.46
规格
10mg; 50mg
规格(数值)
10 mg
别名
3-[4-(Hexyloxy)-1,2,5-thiadiazol-3- yl]-1,2,5,6-tetrahydro-1-methylpyridine oxalate
溶解性
Soluble to 10 mM in water and to 100 mM in DMSO
储存条件
Desiccate at +4°C
销量
0

产品描述

Functionally selective muscarinic M 1 receptor agonist (EC 50 values are 0.3, 5, 42, 52 and 92.5 nM at M 1 , M 3 , M 5 , M 4 and M 2 receptors respectively). Displays a complex pharmacological profile; reversible and wash-resistant binding resulting in full agonist activity at M 1 , delayed wash-resistant partial agonist activity at M 2 and delayed wash-resistant full agonist activity at M 4 . Exhibits antipsychotic activity, and improves cognitive deficits and behavioral disturbances in Alzheimer's disease and schizophrenia. Purity: >98 %

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