

YIL 781
¥0
- 货号
- YIL 781
- CAS 号
- [875258-85-8]
- 分子式
- C 24 H 28 FN 3 O 2 .HCl
- 分子量
- 445.96
- 规格
- 10mg; 50mg
- 规格(数值)
- 10 mg
- 别名
- 6-(4-Fluorophenoxy)-2-methyl-3-[[(3 S)-1-(1-methylethyl)-3-piperidinyl]methyl]-4(3H)-q uinazolinone
- 溶解性
- Soluble to 100 mM in DMSO and to 100 mM in ethanol
- 储存条件
- Desiccate at RT
- 销量
- 0
产品描述
Ghrelin receptor antagonist (GHS-R1a) (K i = 17 nM). Displays no significant affinity for the motilin receptor (K i = 6 μM). Blocks the effects of ghrelin on insulin secretion both in vivo and in vitro. Improves glucose homeostasis in vivo. Purity: >98 %